SCHEMBL8611570

SCHEMBL8611570

COC(=O)c1ccc(OC(F)(F)F)cc1F.NC(N)=NC(=O)c1ccc(OC(F)(F)F)cc1F

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
ABL1 P00519 1/20 0.38
CPS1 P31327 2/20 0.36
PDE2A O00408 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SCN9A Q15858 1/20 0.36
CNR2 P34972 1/20 0.36
CHEK1 O14757 1/20 0.36
PARP14 Q460N5 1/20 0.36
PARP10 Q53GL7 1/20 0.36
EPHX2 P34913 1/20 0.35
PIM1 P11309 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018666 0.92 PIM1 (0.40) PDE2AKMT2ACHEK1PARP10EPHX2
SCHEMBL8610216 0.88 MRGPRX4 (0.39) CFTRMRGPRX4ABL1KMT2AALDH1A1
SCHEMBL20644248 0.87 CFTR (0.46) CFTRMRGPRX4ABL1CPS1PDE2A
SCHEMBL8609955 0.84 CFTR (0.57) CFTRMRGPRX4ALDH1A1KDM4EGAA
SCHEMBL8610122 0.82 SLC9A1 (0.40) CFTRMRGPRX4
SCHEMBL9018732 0.81 FFAR4 (0.40) ABL1KMT2ACHEK1EPHX2PIM1
SCHEMBL8614095 0.81 MRGPRX4 (0.38) CFTRMRGPRX4ABL1CHEK1EPHX2
SCHEMBL8614188 0.81 MRGPRX4 (0.40) CFTRMRGPRX4KMT2AKDM4EGAA
SCHEMBL8612520 0.80 SLC9A1 (0.40) MRGPRX4PDE2A
SCHEMBL8612355 0.78 TDP1 (0.47) MRGPRX4KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5747539-A Fluorine-containing benzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-05-05 US disclosed