SCHEMBL8612757

SCHEMBL8612757

CC(C)OP(=O)(CN(c1cccnc1)c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1)OC(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 4/20 0.42
ALOX5 P09917 2/20 0.41
PTGS2 P35354 2/20 0.41
PTGS1 P23219 1/20 0.41
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
HSP90AA1 P07900 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
MAPK1 P28482 1/20 0.37
MC4R P32245 1/20 0.37
HTT P42858 1/20 0.37
CCR6 P51684 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8611255 0.88 ALOX5 (0.43) HMGCRALOX5PTGS2PTGS1ALDH1A1
SCHEMBL7120195 0.86 HMGCR (0.43) HMGCRALOX5PTGS2PTGS1ALDH1A1
SCHEMBL8583640 0.85 HMGCR (0.35) HMGCRALOX5PTGS2PTGS1KDM4E
SCHEMBL7128467 0.84 ALOX5 (0.46) ALOX5PTGS2PTGS1ALDH1A1LMNA
SCHEMBL7126919 0.84 ERN1 (0.38) KDM4EALDH1A1LMNAMAPTALOX15
SCHEMBL7121061 0.81 ERN1 (0.36) KDM4ELMNAMAPTALOX15CYP3A4
SCHEMBL7129122 0.81 HMGCR (0.38) HMGCRALOX5PTGS2PTGS1ALDH1A1
SCHEMBL7126160 0.78 RAB9A (0.34) KDM4EALDH1A1LMNATP53MAPT
SCHEMBL7130110 0.77 PTAFR (0.35) ALOX5PTGS2PTGS1KDM4EALDH1A1
SCHEMBL7117974 0.76 PTAFR (0.37) ALOX5PTGS2KDM4ECYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835116-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SYMPHAR S.A. (CH) 1998-04-15 EP claimed
WO-1997002037-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SYMPHAR S.A. (CH) 1997-01-23 WO claimed