SCHEMBL8613368

SCHEMBL8613368

COc1ccc(NS(C)(=O)=O)c2c(NC(=N)NC=O)cc(-c3ccccc3C)nc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 4/20 0.38
CCNT1 O60563 1/20 0.36
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
MAPK1 P28482 1/20 0.35
NR3C1 P04150 2/20 0.33
ALPL P05186 2/20 0.33
PTK2 Q05397 3/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
PGR P06401 1/20 0.33
NR3C2 P08235 1/20 0.33
AR P10275 1/20 0.33
TSHR P16473 2/20 0.33
HTT P42858 2/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613234 0.93 CDK9 (0.38) CDK9CCNT1ALDH1A1MEN1KMT2A
SCHEMBL8619171 0.89 MAPT (0.39) ALDH1A1MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL8619262 0.88 BACE1 (0.41) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL8620853 0.88 ADORA3 (0.36) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL8614891 0.85 NQO2 (0.34) MEN1KMT2ASMN1; SMN2POLBMAPT
SCHEMBL8618644 0.85 ADORA3 (0.34) CDK9CCNT1ALDH1A1MEN1KMT2A
SCHEMBL8617517 0.85 MAPT (0.34) ALDH1A1MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL8615517 0.85 ALDH1A1 (0.34) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL8615844 0.84 ADORA3 (0.36) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL8616647 0.83 KDM4E (0.38) PTK2HTTPOLBMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed