SCHEMBL8614754

SCHEMBL8614754

COc1c(OC)c(OC)c2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc2c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.44
PLA2G2A P14555 1/20 0.41
CYP3A4 P08684 2/20 0.40
KDM4E B2RXH2 4/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
MAPT P10636 3/20 0.40
ALOX12 P18054 2/20 0.40
TACR3 P29371 2/20 0.40
HTT P42858 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ALDH1A1 P00352 4/20 0.39
HPGD P15428 4/20 0.39
PPARA Q07869 1/20 0.39
CASP1 P29466 1/20 0.39
MAPK1 P28482 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ALOX5 P09917 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8616466 0.88 PDE10A (0.47) PDE10ACYP3A4KDM4EMEN1KMT2A
SCHEMBL8614027 0.88 PDE10A (0.47) PDE10ACYP3A4KDM4EMEN1KMT2A
SCHEMBL8619690 0.86 TACR3 (0.40) KDM4EMEN1KMT2AMAPTTACR3
SCHEMBL8614344 0.84 PDE10A (0.52) PDE10APLA2G2AKDM4EMEN1KMT2A
SCHEMBL8619812 0.84 ALDH1A1 (0.54) PLA2G2ACYP3A4KDM4EMEN1KMT2A
SCHEMBL8613185 0.84 PDE10A (0.49) PDE10ACYP3A4KDM4EMEN1KMT2A
SCHEMBL8617942 0.82 MEN1 (0.50) PLA2G2ACYP3A4KDM4EMEN1KMT2A
SCHEMBL8614875 0.82 PDE10A (0.52) PDE10ACYP3A4KDM4EMEN1KMT2A
SCHEMBL8617709 0.79 PDE10A (0.69) PDE10ACYP3A4KDM4EMEN1KMT2A
SCHEMBL8620626 0.79 ALDH1A1 (0.48) PDE10APLA2G2ACYP3A4KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed