SCHEMBL8619690

SCHEMBL8619690

COc1c(OC)c(OC)c2c(C(=O)NC(=N)N)cc(-c3ccccc3C)nc2c1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.40
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
HPGD P15428 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HTT P42858 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
GPR55 Q9Y2T6 1/20 0.38
KDM4E B2RXH2 2/20 0.36
SMYD2 Q9NRG4 2/20 0.36
POLB P06746 3/20 0.35
THRB P10828 1/20 0.35
ADORA2A P29274 2/20 0.35
ADORA1 P30542 2/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618478 0.89 THRB (0.39) TACR3CA2CA9CA12CA1
SCHEMBL8616639 0.89 THRB (0.39) TACR3CA2CA9CA12CA1
SCHEMBL8614754 0.86 PDE10A (0.44) TACR3KMT2AMEN1HPGDHTT
SCHEMBL8619166 0.85 TACR3 (0.40) TACR3CA2CA9CA12CA1
SCHEMBL8617847 0.85 TACR3 (0.42) TACR3CA2CA9CA12CA1
SCHEMBL8613206 0.85 ALDH1A1 (0.45) TACR3CA2CA9CA12CA1
SCHEMBL8615841 0.84 TACR3 (0.39) TACR3CA2CA9CA12CA1
SCHEMBL8620849 0.84 TACR3 (0.39) TACR3CA2CA9CA12CA1
SCHEMBL8618016 0.84 CA2 (0.44) TACR3CA2CA9CA12CA1
SCHEMBL8619742 0.84 TACR3 (0.43) TACR3CA2CA9CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed