SCHEMBL8614767

SCHEMBL8614767

COc1c(OC)c(OC)c2c(NC(=N)NC=O)cc(-c3ccccc3)nc2c1OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.36
MAPT P10636 5/20 0.36
HPGD P15428 4/20 0.36
KDM4E B2RXH2 3/20 0.36
CYP2C19 P33261 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
NQO2 P16083 1/20 0.35
TSHR P16473 1/20 0.35
ATM Q13315 1/20 0.35
ADORA3 P0DMS8 3/20 0.35
ALDH1A1 P00352 4/20 0.34
ADORA1 P30542 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
TACR3 P29371 1/20 0.34
ACP1 P24666 1/20 0.33
IDO1 P14902 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614038 0.89 PDE10A (0.39) PDE10AMAPTHPGDKDM4ECYP2C19
SCHEMBL8616478 0.89 PDE10A (0.39) PDE10AMAPTHPGDKDM4ECYP2C19
SCHEMBL8619826 0.86 ALDH1A1 (0.44) MAPTHPGDKDM4ECYP2C19CYP3A4
SCHEMBL8619697 0.86 POLB (0.33) MAPTKDM4EMEN1KMT2AADORA3
SCHEMBL8614352 0.85 PDE10A (0.43) PDE10AMAPTHPGDKDM4EMEN1
SCHEMBL8613198 0.84 PDE10A (0.41) PDE10AMAPTHPGDKDM4ECYP2C19
SCHEMBL8617947 0.84 MEN1 (0.43) MAPTHPGDKDM4ECYP2C19CYP3A4
SCHEMBL8614881 0.82 TDO2 (0.43) PDE10AMAPTHPGDKDM4ECYP2C19
SCHEMBL8620632 0.80 HPGD (0.44) PDE10AMAPTHPGDKDM4ECYP3A4
SCHEMBL8617718 0.80 PDE10A (0.56) PDE10AMAPTHPGDNQO2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed