SCHEMBL8614038

SCHEMBL8614038

COc1cc(OC)c2c(NC(=N)NC=O)cc(-c3ccccc3)nc2c1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.39
HPGD P15428 4/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.36
POLB P06746 2/20 0.36
USP2 O75604 1/20 0.36
HSD17B10 Q99714 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
PDGFRB P09619 1/20 0.36
ACHE P22303 2/20 0.36
ALDH1A1 P00352 2/20 0.36
BACE1 P56817 1/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TACR3 P29371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8616478 0.92 PDE10A (0.39) PDE10AHPGDMAPTKDM4ECYP3A4
SCHEMBL8614352 0.89 PDE10A (0.43) PDE10AHPGDMAPTKDM4EHTT
SCHEMBL8614767 0.89 PDE10A (0.36) PDE10AHPGDMAPTKDM4ECYP3A4
SCHEMBL8618493 0.87 KDM4E (0.38) MAPTKDM4EHTTPOLBUSP2
SCHEMBL8613198 0.86 PDE10A (0.41) PDE10AHPGDMAPTKDM4ECYP3A4
SCHEMBL8614881 0.86 TDO2 (0.43) PDE10AHPGDMAPTKDM4ECYP3A4
SCHEMBL8619826 0.86 ALDH1A1 (0.44) HPGDMAPTKDM4ECYP3A4CYP2C9
SCHEMBL8617947 0.84 MEN1 (0.43) HPGDMAPTKDM4ECYP3A4CYP2C9
SCHEMBL8616318 0.82 BACE1 (0.41) PDE10AHPGDMAPTKDM4ECYP3A4
SCHEMBL8618666 0.82 KDM4E (0.44) HPGDMAPTKDM4ECYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed