SCHEMBL8614898

SCHEMBL8614898

COc1ccc(Br)c2nc(-c3ccccc3C)cc(NC(=N)NC=O)c12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.34
LMNA P02545 2/20 0.33
LTB4R Q15722 1/20 0.33
HPGD P15428 1/20 0.33
ADORA3 P0DMS8 3/20 0.32
MAPT P10636 4/20 0.32
NPC1 O15118 2/20 0.32
GRM4 Q14833 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
KDM4E B2RXH2 3/20 0.31
POLB P06746 2/20 0.31
USP2 O75604 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614891 0.93 NQO2 (0.34) NQO2LMNALTB4RHPGDADORA3
SCHEMBL8619171 0.92 MAPT (0.39) LMNALTB4RADORA3MAPTCA12
SCHEMBL8615844 0.91 ADORA3 (0.36) LMNALTB4RADORA3MAPTKDM4E
SCHEMBL8616041 0.89 ALDH1A1 (0.33) LTB4RADORA3MAPTNPC1KDM4E
SCHEMBL8620853 0.87 ADORA3 (0.36) LMNALTB4RADORA3MAPTKDM4E
SCHEMBL8615517 0.87 ALDH1A1 (0.34) LMNALTB4RADORA3MAPTMEN1
SCHEMBL8618493 0.86 KDM4E (0.38) LMNAADORA3MAPTKDM4EPOLB
SCHEMBL8613234 0.85 CDK9 (0.38) MAPTPOLBMEN1KMT2ASMN1; SMN2
SCHEMBL8617517 0.85 MAPT (0.34) LMNALTB4RADORA3MAPTKDM4E
SCHEMBL8618644 0.85 ADORA3 (0.34) LTB4RADORA3MAPTKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed