SCHEMBL8615313

SCHEMBL8615313

COC(C)Oc1cccc2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.54
TACR3 P29371 11/20 0.45
ACACA Q13085 1/20 0.43
TACR2 P21452 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
TSHR P16473 2/20 0.42
CYP3A4 P08684 2/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP1A2 P05177 1/20 0.42
NFKB1 P19838 1/20 0.42
MTOR P42345 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CCR6 P51684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615930 0.96 PDE10A (0.51) PDE10ATACR3ACACATACR2ALDH1A1
SCHEMBL8617709 0.89 PDE10A (0.69) PDE10AACACAALDH1A1MEN1KMT2A
SCHEMBL8617941 0.85 PDE10A (0.64) PDE10AACACAALDH1A1MEN1KMT2A
SCHEMBL8615321 0.84 PDE10A (0.54) PDE10ATACR3ACACATACR2ALDH1A1
SCHEMBL8613515 0.84 PDE10A (0.76) PDE10AALDH1A1KDM4EHSD17B10CCR6
SCHEMBL8620680 0.84 ALDH1A1 (0.54) PDE10AACACAALDH1A1MEN1KMT2A
SCHEMBL8615931 0.81 PDE10A (0.51) PDE10ATACR3ACACATACR2ALDH1A1
SCHEMBL8613481 0.81 KDM4E (0.56) PDE10AALDH1A1MEN1KMT2ATSHR
SCHEMBL8615990 0.80 CCR6 (0.57) PDE10ATACR3ALDH1A1MEN1KMT2A
SCHEMBL8616695 0.80 MEN1 (0.46) PDE10ATACR3ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed