SCHEMBL8620680

SCHEMBL8620680

CCOc1cccc2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
POLB P06746 2/20 0.54
PDE10A Q9Y233 1/20 0.54
CCR6 P51684 1/20 0.50
ACACA Q13085 2/20 0.47
MEN1 O00255 8/20 0.47
KMT2A Q03164 8/20 0.47
GAA P10253 2/20 0.47
TP53 P04637 2/20 0.46
LMNA P02545 4/20 0.46
KDM4E B2RXH2 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HTT P42858 2/20 0.46
RAB9A P51151 3/20 0.45
NPC1 O15118 2/20 0.44
HPGD P15428 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
ATM Q13315 1/20 0.43
ALOX12 P18054 1/20 0.43
NFKB1 P19838 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615321 0.90 PDE10A (0.54) ALDH1A1POLBPDE10ACCR6ACACA
SCHEMBL8617709 0.89 PDE10A (0.69) ALDH1A1POLBPDE10ACCR6ACACA
SCHEMBL8617400 0.87 MEN1 (0.46) ALDH1A1POLBMEN1KMT2AGAA
SCHEMBL8615931 0.87 PDE10A (0.51) ALDH1A1POLBPDE10ACCR6ACACA
SCHEMBL8617941 0.85 PDE10A (0.64) ALDH1A1POLBPDE10AACACAMEN1
SCHEMBL8615313 0.84 PDE10A (0.54) ALDH1A1PDE10ACCR6ACACAMEN1
SCHEMBL8618650 0.84 LMNA (0.47) ALDH1A1POLBPDE10AMEN1KMT2A
SCHEMBL28184818 0.84 PDE10A (0.75) ALDH1A1POLBPDE10ACCR6ACACA
SCHEMBL8613763 0.83 TACR3 (0.46) ALDH1A1PDE10ACCR6MEN1KMT2A
SCHEMBL8613481 0.83 KDM4E (0.56) ALDH1A1POLBPDE10ACCR6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed