SCHEMBL8615511

SCHEMBL8615511

Cc1ccccc1-c1cc(NC(=N)NC=O)c2ccc(OC3CC3)cc2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 2/20 0.35
ACSL1 P33121 4/20 0.35
ACP1 P24666 2/20 0.35
DNMT1 P26358 1/20 0.34
EHMT2 Q96KQ7 1/20 0.34
PKM P14618 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.33
F2 P00734 1/20 0.33
PLG P00747 1/20 0.33
PRSS1 P07477 1/20 0.33
P2RX7 Q99572 1/20 0.33
ACACB O00763 2/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614075 0.89 CA2 (0.38) TACR3ACSL1ACP1DNMT1EHMT2
SCHEMBL8617721 0.89 CA2 (0.38) TACR3ACSL1ACP1DNMT1EHMT2
SCHEMBL8619346 0.88 TACR3 (0.46) TACR3PKMCA12CA1CA2
SCHEMBL8613388 0.87 SMN1; SMN2 (0.39) TACR3PKMCA12CA1CA2
SCHEMBL8617128 0.86 ACP1 (0.35) TACR3ACP1DNMT1EHMT2PKM
SCHEMBL8613990 0.84 TACR3 (0.39) TACR3ACP1DNMT1EHMT2PKM
SCHEMBL8615573 0.83 TACR3 (0.37) TACR3ACP1DNMT1EHMT2PKM
SCHEMBL8615853 0.83 TACR3 (0.37) TACR3PKMCA12CA1CA2
SCHEMBL8620107 0.83 HTT (0.37) TACR3ACP1CA12CA1CA2
SCHEMBL8620892 0.82 HTT (0.47) TACR3ACP1MEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed