SCHEMBL8615747

SCHEMBL8615747

CN1CCN(c2ccc3c(=O)cc[nH]c3c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
HSD17B10 Q99714 2/20 0.44
MAP3K11 Q16584 1/20 0.43
KIF11 P52732 2/20 0.43
HTR3A P46098 1/20 0.43
ERCC1 P07992 1/20 0.43
DNASE1 P24855 1/20 0.43
FEN1 P39748 1/20 0.43
ERCC4 Q92889 1/20 0.43
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42
PTK2B Q14289 1/20 0.42
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29576625 1.00 ALDH1A1 (0.49) ALDH1A1HSD17B10MAP3K11KIF11HTR3A
SCHEMBL28826859 0.84 PIK3CD (0.53) ALDH1A1HSD17B10MAP3K11KIF11ERCC1
SCHEMBL29576228 0.84 ALDH1A1 (0.50) ALDH1A1HSD17B10HTR3AERCC1DNASE1
SCHEMBL7291426 0.84 ALDH1A1 (0.50) ALDH1A1HSD17B10HTR3AERCC1DNASE1
SCHEMBL5097444 0.80 HTR3A (0.57) ALDH1A1HSD17B10HTR3AGAAKDM4E
SCHEMBL9569216 0.78 ALDH1A1 (0.44) ALDH1A1HSD17B10MAP3K11ERCC1DNASE1
SCHEMBL9569202 0.78 ALDH1A1 (0.41) ALDH1A1HSD17B10MAP3K11ERCC1DNASE1
SCHEMBL20443487 0.77 HTR3A (0.50) ALDH1A1HSD17B10HTR3AGAAKDM4E
SCHEMBL949366 0.75 HTR3A (0.56) HTR3AGAAKDM4EMAPTMAPK1
SCHEMBL18436001 0.74 ADRA2C (0.47) ALDH1A1HSD17B10HTR3AGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831845-A4 DIPHOSPHONATE DERIVATIVES OF THERAPEUTIC AGENTS ELIZANOR BIOPHARMACEUTICALS IN (US) 1998-12-02 EP claimed
EP-0831845-A1 DIPHOSPHONATE DERIVATIVES OF THERAPEUTIC AGENTS Elizanor Biopharmaceuticals, Inc. (US) 1998-04-01 EP claimed
WO-1996040156-A1 DIPHOSPHONATE DERIVATIVES OF THERAPEUTIC AGENTS ELIZANOR BIOPHARMACEUTICALS, INC. (US) 1996-12-19 WO claimed