SCHEMBL8616494

SCHEMBL8616494

CC(C)C(C)Cc1ccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c2c1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 2/20 0.39
NQO2 P16083 1/20 0.39
DHODH Q02127 1/20 0.39
TACR3 P29371 4/20 0.38
MOK Q9UQ07 2/20 0.37
ABCB1 P08183 1/20 0.36
ABCC1 P33527 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
CACNA2D1 P54289 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615126 0.90 DHODH (0.47) ACP1DHODHMOKABCB1ABCC1
SCHEMBL8616641 0.87 ACP1 (0.42) ACP1NQO2DHODHTACR3MOK
SCHEMBL8619039 0.85 DHODH (0.46) ACP1NQO2DHODHTACR3MOK
SCHEMBL8614052 0.84 CACNA2D1 (0.38) ACP1NQO2DHODHTACR3ABCB1
SCHEMBL8619222 0.83 DHODH (0.45) ACP1NQO2DHODHTACR3MOK
SCHEMBL8615306 0.83 TACR3 (0.42) ACP1NQO2DHODHTACR3MOK
SCHEMBL8614060 0.83 DHODH (0.44) ACP1NQO2DHODHTACR3ABCB1
SCHEMBL8617746 0.81 TACR3 (0.41) ACP1NQO2DHODHTACR3MOK
SCHEMBL8613853 0.81 ALDH1A1 (0.52) ACP1ABCB1ABCC1ABCG2
SCHEMBL8615684 0.80 ESR1 (0.43) ACP1TACR3ABCB1ABCC1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed