SCHEMBL8615684

SCHEMBL8615684

N=C(NC=O)Nc1cc(-c2ccccc2)nc2ccc(O)cc12

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.43
ESR2 Q92731 9/20 0.43
ESRRB O95718 6/20 0.43
ESRRA P11474 6/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GFER P55789 1/20 0.40
ACP1 P24666 1/20 0.40
ELANE P08246 1/20 0.40
POLB P06746 1/20 0.40
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
TACR3 P29371 1/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615210 0.92 TACR3 (0.44) ESR1ESR2MEN1KMT2AGFER
SCHEMBL8620932 0.88 POLB (0.51) MEN1KMT2AGFERACP1POLB
SCHEMBL8617753 0.88 ACP1 (0.51) MEN1KMT2AGFERACP1ABCB1
SCHEMBL8617521 0.87 TLR9 (0.41) MEN1KMT2AGFERACP1ABCB1
SCHEMBL8617812 0.87 MAPK1 (0.46) MEN1KMT2AACP1
SCHEMBL8615496 0.87 DHODH (0.50) MEN1KMT2AGFERACP1ABCB1
SCHEMBL8614838 0.87 MEN1 (0.40) MEN1KMT2AGFERACP1ABCB1
SCHEMBL8613853 0.87 ALDH1A1 (0.52) MEN1KMT2AACP1ABCB1ABCC1
SCHEMBL8614861 0.86 AKR1C3 (0.53) MEN1KMT2AGFERACP1ABCB1
SCHEMBL8614948 0.85 HTT (0.39) ESR1ESR2ESRRBESRRAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed