SCHEMBL8613853

SCHEMBL8613853

Cc1ccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
KDM4E B2RXH2 5/20 0.52
HSD17B10 Q99714 1/20 0.52
MAPT P10636 6/20 0.47
LMNA P02545 5/20 0.47
NPSR1 Q6W5P4 4/20 0.47
HPGD P15428 3/20 0.47
HSP90AA1 P07900 3/20 0.47
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
RECQL P46063 1/20 0.46
THRB P10828 3/20 0.46
CYP3A4 P08684 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PDE10A Q9Y233 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617739 0.92 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10MAPTLMNA
SCHEMBL8615355 0.88 PDE10A (0.55) ALDH1A1KDM4EMAPTNPSR1HPGD
SCHEMBL8615684 0.87 ESR1 (0.43) KMT2AMEN1CYP3A4ACP1ABCB1
SCHEMBL8617753 0.87 ACP1 (0.51) KDM4ELMNAKMT2AMEN1CYP3A4
SCHEMBL8618948 0.86 MEN1 (0.50) ALDH1A1KDM4EMAPTLMNAHPGD
SCHEMBL8614838 0.86 MEN1 (0.40) KDM4ELMNAKMT2AMEN1CYP3A4
SCHEMBL8617812 0.86 MAPK1 (0.46) ALDH1A1KDM4EHSD17B10MAPTLMNA
SCHEMBL8617521 0.86 TLR9 (0.41) ALDH1A1KDM4EMAPTLMNAHPGD
SCHEMBL8615496 0.86 DHODH (0.50) ALDH1A1KMT2AMEN1CYP3A4GAA
SCHEMBL8620945 0.85 NQO2 (0.56) ALDH1A1KDM4EKMT2AMEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed