SCHEMBL8614060

SCHEMBL8614060

CC(C)c1ccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c2c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.44
TP53 P04637 3/20 0.41
MAPT P10636 1/20 0.41
ACP1 P24666 1/20 0.40
TACR3 P29371 2/20 0.39
PTGFR P43088 1/20 0.39
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ADORA1 P30542 1/20 0.38
NQO2 P16083 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619401 0.87 ABCB1 (0.44) DHODHACP1TACR3ABCB1ABCC1
SCHEMBL8613853 0.85 ALDH1A1 (0.52) MAPTACP1ABCB1ABCC1ABCG2
SCHEMBL8615684 0.84 ESR1 (0.43) ACP1TACR3ABCB1ABCC1ABCG2
SCHEMBL8617753 0.84 ACP1 (0.51) ACP1ABCB1ABCC1ABCG2SMN1; SMN2
SCHEMBL8614838 0.83 MEN1 (0.40) ACP1PTGFRABCB1ABCC1ABCG2
SCHEMBL8615496 0.83 DHODH (0.50) DHODHACP1ABCB1ABCC1ABCG2
SCHEMBL8617521 0.83 TLR9 (0.41) MAPTACP1ABCB1ABCC1ABCG2
SCHEMBL8617812 0.83 MAPK1 (0.46) DHODHMAPTACP1HPGDMEN1
SCHEMBL8620945 0.83 NQO2 (0.56) ACP1TACR3ABCB1ABCG2SMN1; SMN2
SCHEMBL8613674 0.83 TRPV1 (0.43) MAPTACP1TACR3PTGFRABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed