SCHEMBL8616713

SCHEMBL8616713

CS(=O)(=O)Oc1ccc(C[C@@H](CNCCN)NC(=O)OCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.50
ITGB3 P05106 7/20 0.49
ITGA2B P08514 7/20 0.49
PPARG P37231 2/20 0.46
CTSL P07711 2/20 0.44
CTSK P43235 2/20 0.44
SYK P43405 1/20 0.44
P2RX7 Q99572 3/20 0.44
ATM Q13315 1/20 0.43
PPARA Q07869 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8615937 0.99 CTRB1 (0.49) CTRB1ITGB3ITGA2BPPARGCTSL
SCHEMBL8611915 0.86 ITGB3 (0.56) CTRB1ITGB3ITGA2B
Hydrochloric Acid SCHEMBL8612059 0.85 ITGB3 (0.55) CTRB1ITGB3ITGA2B
SCHEMBL1823130 0.83 CTRB1 (0.55) CTRB1ITGB3ITGA2BPPARGCTSL
SCHEMBL1823016 0.82 CTRB1 (0.54) CTRB1ITGB3ITGA2BPPARGCTSL
SCHEMBL1824729 0.80 CTRB1 (0.52) CTRB1ITGB3ITGA2BPPARGSYK
SCHEMBL1825873 0.79 CTRB1 (0.51) CTRB1ITGB3ITGA2BPPARGCTSL
SCHEMBL5158241 0.79 CTRB1 (0.53) CTRB1ITGB3ITGA2BCTSLCTSK
SCHEMBL1824337 0.78 SYK (0.53) CTRB1ITGB3ITGA2BPPARGCTSL
SCHEMBL1825917 0.78 ALDH1A1 (0.58) ITGB3ITGA2BPPARGCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680467-B1 PROCESS FOR PREPARING C-SUBSTITUTED DIETHYLENE TRIAMINES SCHERING AG (DE) 1998-04-22 EP disclosed
US-5654467-A Process for the production of C-substituted diethylenetriamines SCHERING AKTIENGESELLSCHAFT (DE) 1997-08-05 US disclosed
EP-0680467-A1 PROCESS FOR PREPARING C-SUBSTITUTED DIETHYLENE TRIAMINES SCHERING AKTIENGESELLSCHAFT (DE) 1995-11-08 EP disclosed
WO-1994017033-A1 PROCESS FOR PREPARING C-SUBSTITUTED DIETHYLENE TRIAMINES SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-04 WO disclosed