SCHEMBL8779130

SCHEMBL8779130

O=C(O)c1cc(C(=O)O)cc(-c2ccc(F)c(Cl)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 3/20 0.55
RPA1 P27694 1/20 0.54
RXRA P19793 2/20 0.50
RXRB P28702 2/20 0.50
ERCC1 P07992 1/20 0.50
ERCC4 Q92889 1/20 0.50
CASP1 P29466 1/20 0.47
DHODH Q02127 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HSD17B1 P14061 1/20 0.45
HSD17B2 P37059 1/20 0.45
TPMT P51580 1/20 0.45
MARS1 P56192 1/20 0.45
ICMT O60725 1/20 0.45
ACLY P53396 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
HSD17B14 Q9BPX1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3643412 0.87 RXRA (0.61) KMORPA1RXRARXRBERCC1
Biguanide SCHEMBL8617033 0.87 KMO (0.45) KMORPA1RXRARXRBERCC1
SCHEMBL30308290 0.79 TSHR (0.65) KMORPA1RXRARXRBKDM4E
SCHEMBL109599 0.79 TSHR (0.65) KMORPA1RXRARXRBKDM4E
SCHEMBL16608990 0.79 RPA1 (0.58) KMORPA1ERCC1ERCC4CASP1
SCHEMBL11693280 0.78 AKR1C2 (0.66) KMORPA1ERCC1ERCC4CASP1
Hydrochloric Acid SCHEMBL7105574 0.77 TSHR (0.63) KMORPA1RXRARXRBKDM4E
SCHEMBL3979148 0.76 ACMSD (0.59) KMORPA1ERCC1ERCC4KDM4E
SCHEMBL15814719 0.76 DHODH (0.69) KMORXRARXRBDHODH
SCHEMBL16488615 0.76 DHODH (0.69) KMORXRARXRBDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0774457-A1 Substituted benzodicarboxylic acid diguanidines, process for their preparation, and their use as medicament or diagnostic agent HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-21 EP disclosed