SCHEMBL8620212

SCHEMBL8620212

N=C(NC=O)Nc1cc(-c2ccccc2)nc2cc(NS(=O)(=O)C3CCCC3)ccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SGK1 O00141 1/20 0.38
BRD4 O60885 2/20 0.37
MAP2K4 P45985 2/20 0.37
AAK1 Q2M2I8 6/20 0.37
GAK O14976 2/20 0.37
STK16 O75716 2/20 0.37
BMP2K Q9NSY1 2/20 0.37
ACP1 P24666 3/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
ACLY P53396 1/20 0.36
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
TACR3 P29371 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HSP90AA1 P07900 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615149 0.85 ALDH1A1 (0.49) ACP1ABCB1ABCC1ABCG2TACR3
SCHEMBL8617822 0.82 ACLY (0.38) ACP1ACLYABCB1ABCC1ABCG2
SCHEMBL8617828 0.81 DHODH (0.45) ACP1ABCB1ABCC1ABCG2TACR3
SCHEMBL8613247 0.81 ALDH1A1 (0.44) ACP1ABCB1ABCC1ABCG2TACR3
SCHEMBL8618955 0.81 ACLY (0.41) AAK1GAKSTK16BMP2KACP1
SCHEMBL8619887 0.81 DHODH (0.47) ACP1ABCB1ABCC1ABCG2TACR3
SCHEMBL8618223 0.80 ALDH1A1 (0.41) AAK1GAKSTK16BMP2KACP1
SCHEMBL8612679 0.80 ABCB1 (0.55) ABCB1ABCC1ABCG2TACR3KDM4E
SCHEMBL8619389 0.79 TACR3 (0.41) ACP1ABCB1ABCC1ABCG2TACR3
SCHEMBL8613743 0.78 ALDH1A1 (0.53) ABCB1ABCC1ABCG2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed