SCHEMBL8617844

SCHEMBL8617844

N=C(N)NC(=O)c1nccc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.55
HDAC6 Q9UBN7 3/20 0.49
HDAC3 O15379 2/20 0.49
HDAC4 P56524 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC7 Q8WUI4 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC10 Q969S8 2/20 0.49
HDAC11 Q96DB2 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC9 Q9UKV0 2/20 0.49
HDAC5 Q9UQL6 2/20 0.49
CNR2 P34972 5/20 0.49
MAPT P10636 2/20 0.48
MEN1 O00255 1/20 0.48
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
KMT2A Q03164 1/20 0.48
PLAU P00749 2/20 0.44
PLG P00747 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5655604 0.82 RAB9A (0.62) RAB9AHDAC6HDAC3HDAC4HDAC1
SCHEMBL2230478 0.80 RAB9A (0.60) RAB9AHDAC6HDAC3HDAC4HDAC1
SCHEMBL111310 0.80 CNR2 (0.53) RAB9AHDAC6HDAC3HDAC4HDAC1
SCHEMBL29358323 0.80 CNR2 (0.53) RAB9AHDAC6HDAC3HDAC4HDAC1
SCHEMBL25474761 0.79 RAB9A (0.58) RAB9AHDAC6HDAC3HDAC4HDAC1
SCHEMBL13306750 0.79 RAB9A (0.58) RAB9AHDAC6HDAC3HDAC4HDAC1
SCHEMBL30956107 0.79 RAB9A (0.58) RAB9AHDAC6HDAC3HDAC4HDAC1
Hydrochloric Acid SCHEMBL4433615 0.78 CNR2 (0.51) RAB9AHDAC6HDAC3HDAC4HDAC1
Naphthalene SCHEMBL10758679 0.78 CNR2 (0.51) RAB9AHDAC6HDAC3HDAC4HDAC1
SCHEMBL28198741 0.78 CNR2 (0.51) RAB9AHDAC6HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed
US-5416094-A Antiarrhythmic and cardioprotective substituted -1(2H)isoquinolines, medicament containing them, and their use for combating heart failures HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-16 US disclosed