SCHEMBL8617855

SCHEMBL8617855

CCCCc1cccc2nc(-c3ccccc3)cc(C(=O)NC(=N)N)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.47
TACR3 P29371 7/20 0.46
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PLA2G2A P14555 1/20 0.42
TSHR P16473 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
CYP2C9 P11712 1/20 0.42
TACR2 P21452 2/20 0.41
PTGER4 P35408 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KCNH2 Q12809 2/20 0.41
HPGD P15428 1/20 0.41
CYP1A2 P05177 1/20 0.41
ALOX12 P18054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615443 0.89 ALDH1A1 (0.42) DHODHTACR3ALDH1A1TSHRCYP2C9
SCHEMBL8618932 0.82 PTGER4 (0.55) DHODHTACR3KDM4EALDH1A1LMNA
SCHEMBL8615259 0.81 TACR3 (0.42) DHODHTACR3KDM4EALDH1A1LMNA
SCHEMBL8614299 0.81 DHODH (0.48) DHODHTACR3KDM4EALDH1A1GAA
SCHEMBL8618650 0.81 LMNA (0.47) TACR3KDM4EALDH1A1LMNAGAA
SCHEMBL8613359 0.81 MEN1 (0.46) DHODHTACR3KDM4EALDH1A1LMNA
SCHEMBL8617715 0.81 MEN1 (0.46) DHODHTACR3KDM4EALDH1A1LMNA
SCHEMBL8615669 0.80 TACR3 (0.47) DHODHTACR3KDM4EALDH1A1LMNA
SCHEMBL8619780 0.80 ADORA3 (0.47) TACR3KDM4EALDH1A1LMNAGAA
SCHEMBL8616258 0.80 MEN1 (0.46) DHODHTACR3KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed