SCHEMBL8619780

SCHEMBL8619780

CCC(=O)Nc1cccc2nc(-c3ccccc3)cc(C(=O)NC(=N)N)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.47
ADORA2A P29274 2/20 0.47
ADORA2B P29275 2/20 0.47
ADORA1 P30542 2/20 0.47
MEN1 O00255 6/20 0.46
KMT2A Q03164 6/20 0.46
ALDH1A1 P00352 5/20 0.46
CYP3A4 P08684 3/20 0.46
CYP1A2 P05177 2/20 0.46
ALOX12 P18054 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 2/20 0.46
IKBKB O14920 1/20 0.45
GFER P55789 1/20 0.44
KDM4E B2RXH2 3/20 0.44
HPGD P15428 2/20 0.44
MAPT P10636 1/20 0.44
PTGER4 P35408 1/20 0.43
KCNH2 Q12809 2/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614054 0.89 KMT2A (0.51) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL8618116 0.86 ADORA1 (0.47) ADORA3ADORA2AADORA1MEN1KMT2A
SCHEMBL8614946 0.85 ALDH1A1 (0.43) MEN1KMT2AALDH1A1CYP3A4CYP1A2
SCHEMBL8615326 0.83 MEN1 (0.45) MEN1KMT2AALDH1A1CYP3A4CYP1A2
SCHEMBL8618932 0.82 PTGER4 (0.55) MEN1KMT2AALDH1A1CYP3A4CYP1A2
SCHEMBL8615259 0.81 TACR3 (0.42) MEN1KMT2AALDH1A1CYP3A4CYP1A2
SCHEMBL8618650 0.81 LMNA (0.47) MEN1KMT2AALDH1A1CYP3A4CYP1A2
SCHEMBL8617715 0.81 MEN1 (0.46) MEN1KMT2AALDH1A1CYP3A4CYP1A2
SCHEMBL8613359 0.81 MEN1 (0.46) MEN1KMT2AALDH1A1CYP3A4CYP1A2
SCHEMBL8617855 0.80 DHODH (0.47) MEN1KMT2AALDH1A1CYP1A2ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed