SCHEMBL8618655

SCHEMBL8618655

CCOc1cccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.45
TP53 P04637 3/20 0.41
MAPT P10636 4/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
GAA P10253 1/20 0.40
ACP1 P24666 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ABCB1 P08183 2/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
ABCC1 P33527 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8620632 0.89 HPGD (0.44) PDE10ATP53MAPTMEN1KMT2A
SCHEMBL8615341 0.87 MEN1 (0.39) PDE10ATP53MAPTMEN1KMT2A
SCHEMBL8620687 0.84 PDE10A (0.45) PDE10ATP53MAPTMEN1KMT2A
SCHEMBL8618937 0.83 PTGER4 (0.46) PDE10AMEN1KMT2AACP1ALDH1A1
SCHEMBL8619792 0.82 ADORA1 (0.47) TP53MAPTMEN1KMT2AACP1
SCHEMBL8617724 0.82 ABCG2 (0.41) PDE10AMEN1KMT2AACP1KDM4E
SCHEMBL8617861 0.81 DHODH (0.42) PDE10AACP1ABCB1ABCG2ABCC1
SCHEMBL8614953 0.81 ALDH1A1 (0.42) MAPTMEN1KMT2AACP1ALDH1A1
SCHEMBL8616263 0.81 ABCB1 (0.40) PDE10AMAPTMEN1KMT2AACP1
SCHEMBL8616598 0.81 ABCG2 (0.40) PDE10AMEN1KMT2AACP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed