SCHEMBL8619792

SCHEMBL8619792

CCC(=O)Nc1cccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.47
ADORA3 P0DMS8 2/20 0.47
ADORA2A P29274 2/20 0.47
ADORA2B P29275 2/20 0.47
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
ACP1 P24666 1/20 0.39
ATM Q13315 1/20 0.39
MOK Q9UQ07 2/20 0.38
USP2 O75604 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614064 0.89 ABCB1 (0.50) ADORA1ADORA3ADORA2AADORA2BMEN1
SCHEMBL8618123 0.86 ADORA1 (0.47) ADORA1ADORA3ADORA2AMEN1KMT2A
SCHEMBL8614953 0.85 ALDH1A1 (0.42) ADORA1ADORA3ADORA2AADORA2BMEN1
SCHEMBL8618937 0.83 PTGER4 (0.46) MEN1KMT2AKDM4EALDH1A1ABCB1
SCHEMBL8615331 0.83 ALDH1A1 (0.41) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL8618655 0.82 PDE10A (0.45) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL8617724 0.82 ABCG2 (0.41) MEN1KMT2AKDM4EABCB1ABCC1
SCHEMBL8615265 0.81 MRGPRX1 (0.37) ADORA1ALDH1A1HPGDABCB1ABCC1
SCHEMBL8617861 0.81 DHODH (0.42) ADORA1ABCB1ABCC1ABCG2ACP1
SCHEMBL8613362 0.81 ACHE (0.41) MEN1KMT2AKDM4EABCB1ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed