SCHEMBL8618937

SCHEMBL8618937

Cc1cccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 2/20 0.46
ABCB1 P08183 1/20 0.42
ABCC1 P33527 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
KMT2A Q03164 4/20 0.41
CYP3A4 P08684 3/20 0.41
MEN1 O00255 3/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
ALOX12 P18054 1/20 0.41
CYP2C19 P33261 1/20 0.41
ACP1 P24666 2/20 0.41
TRPV1 Q8NER1 1/20 0.39
PDE10A Q9Y233 2/20 0.37
GFER P55789 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8620877 0.89 HTT (0.39) PTGER4KMT2ACYP3A4MEN1ALDH1A1
SCHEMBL8617724 0.87 ABCG2 (0.41) PTGER4ABCB1ABCC1ABCG2KMT2A
SCHEMBL8616263 0.86 ABCB1 (0.40) PTGER4ABCB1ABCC1ABCG2KMT2A
SCHEMBL8616598 0.86 ABCG2 (0.40) PTGER4ABCB1ABCC1ABCG2KMT2A
SCHEMBL8613362 0.86 ACHE (0.41) PTGER4ABCB1ABCC1ABCG2KMT2A
SCHEMBL8620632 0.86 HPGD (0.44) ABCB1ABCC1ABCG2KMT2ACYP3A4
SCHEMBL8614064 0.86 ABCB1 (0.50) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8615331 0.84 ALDH1A1 (0.41) PTGER4ABCB1ABCC1ABCG2KMT2A
SCHEMBL8615866 0.84 ABCB1 (0.39) PTGER4ABCB1ABCC1ABCG2KMT2A
SCHEMBL8617753 0.83 ACP1 (0.51) ABCB1ABCC1ABCG2KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed