SCHEMBL8618902

SCHEMBL8618902

Cc1ccccc1-c1cc(NC(=N)NC=O)c2cccc(OCOCC(C)C)c2n1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.32
ADORA2A P29274 1/20 0.31
USP2 O75604 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
CYP3A4 P08684 1/20 0.30
BDKRB2 P30411 1/20 0.30
SLC2A1 P11166 1/20 0.30
ACP1 P24666 1/20 0.30
ACACA Q13085 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA2 P47869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617403 0.87 KMT2A (0.41) ADORA2AMAPTMEN1KMT2A
SCHEMBL8617986 0.86 KDM4E (0.32) TACR3USP2MAPTHTTMEN1
SCHEMBL8615146 0.85 ALDH1A1 (0.41) HTTMEN1KMT2A
SCHEMBL8617193 0.84 GAA (0.39) KMT2A
SCHEMBL8613400 0.84 GFER (0.41) MAPTHTTSLC2A1ACP1MEN1
SCHEMBL8617850 0.84 S1PR5 (0.37)
SCHEMBL8620017 0.84 DHODH (0.37) TACR3MAPTHTTACP1MEN1
SCHEMBL8614073 0.83 S1PR5 (0.37)
SCHEMBL8620384 0.82 MCHR1 (0.36) MEN1KMT2AGABRG2GABRB3GABRA2
SCHEMBL8620190 0.82 MEN1 (0.33) TACR3MAPTHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed