SCHEMBL8618911

SCHEMBL8618911

COc1cc(C)cc2c(NC(=N)NC=O)cc(-c3ccccc3C)nc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.34
ADORA3 P0DMS8 5/20 0.33
KMT2A Q03164 2/20 0.33
ADORA1 P30542 2/20 0.33
DNMT1 P26358 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
PDE2A O00408 1/20 0.33
PDE10A Q9Y233 1/20 0.33
MEN1 O00255 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
TACR3 P29371 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
POLB P06746 1/20 0.32
ACP1 P24666 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615214 0.91 PDE2A (0.38) ADORA3KMT2AADORA1PDE2APDE10A
SCHEMBL8613400 0.89 GFER (0.41) KMT2APDE10AMEN1KDM4EPOLB
SCHEMBL8617853 0.87 KDM4E (0.38) C5AR1ADORA3KMT2AADORA1DNMT1
SCHEMBL8619965 0.85 ADORA3 (0.37) ADORA3KMT2AADORA1MEN1CA12
SCHEMBL8618956 0.84 CA12 (0.36) ADORA3KMT2AADORA1DNMT1EHMT2
SCHEMBL8617890 0.84 MEN1 (0.45) C5AR1ADORA3KMT2ADNMT1EHMT2
SCHEMBL8619171 0.84 MAPT (0.39) ADORA3KMT2AADORA1MEN1CA12
SCHEMBL8616647 0.83 KDM4E (0.38) ADORA3ADORA1KDM4EUSP2POLB
SCHEMBL8619745 0.83 CYP1A2 (0.34) ADORA3KMT2AADORA1MEN1CA12
SCHEMBL8615844 0.83 ADORA3 (0.36) ADORA3KMT2AADORA1MEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed