SCHEMBL8615214

SCHEMBL8615214

COc1cc(OC)c2nc(-c3ccccc3C)cc(NC(=N)NC=O)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.38
PDE6D O43924 1/20 0.38
PDE6A P16499 1/20 0.38
PDE6G P18545 1/20 0.38
PDE6B P35913 1/20 0.38
PDE6C P51160 1/20 0.38
PDE6H Q13956 1/20 0.38
PDE10A Q9Y233 1/20 0.38
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
ALDH1A1 P00352 3/20 0.35
CYP1A2 P05177 2/20 0.35
LMNA P02545 2/20 0.35
TSHR P16473 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618911 0.91 C5AR1 (0.34) PDE2APDE10ACA2CA9CA12
SCHEMBL8613400 0.88 GFER (0.41) PDE10AALDH1A1LMNAMEN1KMT2A
SCHEMBL8616302 0.87 PDE10A (0.43) PDE10AALDH1A1LMNACYP3A4MEN1
SCHEMBL8617853 0.86 KDM4E (0.38) CYP1A2LMNATSHRCYP3A4CYP2D6
SCHEMBL8620380 0.85 CA2 (0.39) PDE2APDE6DPDE6APDE6GPDE6B
SCHEMBL8619965 0.85 ADORA3 (0.37) CA2CA9CA12CA1CYP1A2
SCHEMBL8616673 0.84 CA2 (0.50) CA2CA9CA12CA1MEN1
SCHEMBL8619171 0.83 MAPT (0.39) CA2CA9CA12CA1ALDH1A1
SCHEMBL8617890 0.83 MEN1 (0.45) CA2CA9CA12CA1ALDH1A1
SCHEMBL8616647 0.83 KDM4E (0.38) LMNANPSR1MAPTPOLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed