SCHEMBL8619745

SCHEMBL8619745

COc1c(C)ccc2c(NC(=N)NC=O)cc(-c3ccccc3C)nc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.34
CLK4 Q9HAZ1 3/20 0.34
ADORA3 P0DMS8 3/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
CYP2C19 P33261 3/20 0.34
USP2 O75604 2/20 0.34
ALDH1A1 P00352 1/20 0.34
APEX1 P27695 1/20 0.34
CASP7 P55210 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
SMYD2 Q9NRG4 1/20 0.33
TACR3 P29371 1/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
THRB P10828 1/20 0.33
CYP2D6 P10635 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619965 0.92 ADORA3 (0.37) CYP1A2ADORA3ADORA2AADORA2BCYP2C19
SCHEMBL8617853 0.88 KDM4E (0.38) CYP1A2ADORA3ADORA2AADORA2BCYP2C19
SCHEMBL8613400 0.86 GFER (0.41) ALDH1A1APEX1KDM4EPOLBMEN1
SCHEMBL8619697 0.85 POLB (0.33) ADORA3ADORA2AADORA2BUSP2CA12
SCHEMBL8618017 0.84 CA2 (0.36) CYP1A2ADORA3ADORA2AADORA2BCYP2C19
SCHEMBL8615227 0.84 MAPT (0.33) CYP1A2CLK4CYP2C19ALDH1A1CA12
SCHEMBL8618911 0.83 C5AR1 (0.34) ADORA3ADORA2AADORA2BUSP2CA12
SCHEMBL8616305 0.82 MEN1 (0.36) CYP1A2CYP2C19USP2ALDH1A1TACR3
SCHEMBL8616647 0.82 KDM4E (0.38) ADORA3ADORA2AADORA2BUSP2KDM4E
SCHEMBL8615214 0.82 PDE2A (0.38) CYP1A2CLK4ADORA3CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed