SCHEMBL8618920

SCHEMBL8618920

Cc1cc(Cl)cc2c(NC(=N)NC=O)cc(-c3ccccc3)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.39
FABP3 P05413 2/20 0.39
FABP4 P15090 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
FABP5 Q01469 1/20 0.39
PPARA Q07869 1/20 0.38
ABCB1 P08183 1/20 0.36
ABCC1 P33527 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
ADORA3 P0DMS8 2/20 0.35
ACP1 P24666 1/20 0.35
PTGER4 P35408 1/20 0.34
MEN1 O00255 2/20 0.34
MAPT P10636 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPK1 P28482 1/20 0.34
ADORA1 P30542 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613487 0.86 KDM4E (0.44) CYP2C9CYP3A4ABCB1ABCC1ABCG2
SCHEMBL8617812 0.82 MAPK1 (0.46) CYP2C9FABP3FABP4ADORA3ACP1
SCHEMBL8618767 0.81 MAPT (0.40) CYP2C9CYP3A4CYP2D6PPARAABCB1
SCHEMBL8613198 0.79 PDE10A (0.41) CYP2C9CYP3A4ACP1MEN1MAPT
SCHEMBL8619389 0.79 TACR3 (0.41) CYP2C9ABCB1ABCC1ABCG2ADORA3
SCHEMBL8617753 0.78 ACP1 (0.51) CYP3A4ABCB1ABCC1ABCG2ACP1
SCHEMBL8615997 0.78 CCR6 (0.45) CYP2C9CYP3A4ABCB1ABCC1ABCG2
SCHEMBL8613853 0.78 ALDH1A1 (0.52) CYP2C9CYP3A4ABCB1ABCC1ABCG2
SCHEMBL8616302 0.77 PDE10A (0.43) CYP3A4ABCB1ABCG2ADORA3MEN1
SCHEMBL8616699 0.77 ACP1 (0.39) CYP2C9CYP3A4ABCB1ABCC1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed