SCHEMBL8619349

SCHEMBL8619349

CC(=O)N(CC(C)C(=O)OCc1ccccc1)N1CCC[C@@H](CCc2ccncc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACE2 Q9BYF1 1/20 0.36
CYP2C9 P11712 2/20 0.35
CYP2D6 P10635 1/20 0.35
GRIN2B Q13224 1/20 0.35
PREP P48147 2/20 0.35
ACHE P22303 1/20 0.35
FKBP1A P62942 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CTSK P43235 2/20 0.33
CTSL P07711 1/20 0.33
AADAT Q8N5Z0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365778 0.89 ITGB3 (0.45) ACE2FKBP1A
SCHEMBL8103481 0.88 ITGB3 (0.35) ACHECYP19A1
SCHEMBL7371949 0.83 ACE (0.35) CYP2C9CYP2D6ACHECYP19A1CYP3A4
SCHEMBL8619473 0.81 FAAH (0.30)
Hydrochloric Acid SCHEMBL7368927 0.80 ITGB3 (0.34)
SCHEMBL8620398 0.78 MC4R (0.33) CYP19A1
SCHEMBL7374011 0.78 DPP4 (0.36) ACHECYP19A1
SCHEMBL8621139 0.77 ITGB3 (0.37)
Hydrochloric Acid SCHEMBL8619234 0.77 ITGB3 (0.36)
SCHEMBL8621118 0.76 ITGB3 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852045-A Fibrinogen receptor antagonists MERCK & CO., INC. (US) 1998-12-22 US disclosed
US-5502165-A AMIDATION OF CARBOXY COMPOOUND WITH AMINE IN WATER AND SOLVENT MERCK & CO., INC. (US) 1996-03-26 US disclosed