SCHEMBL8103481

SCHEMBL8103481

CC(=O)N(C[C@@H](C)C(=O)O)N1CCC[C@@H](CCc2ccncc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
HRH3 Q9Y5N1 2/20 0.34
CYP19A1 P11511 2/20 0.34
ACE P12821 3/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
ACHE P22303 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
FAAH O00519 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
GFER P55789 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7368927 0.88 ITGB3 (0.34) ITGB3ITGA2B
SCHEMBL8619349 0.88 ACE2 (0.36) CYP19A1ACHE
SCHEMBL8621118 0.87 ITGB3 (0.49) ITGB3ITGA2B
SCHEMBL8622174 0.84 ENO1 (0.33) CYP19A1
SCHEMBL8619473 0.82 FAAH (0.30) ITGB3ITGA2BFAAH
SCHEMBL7341454 0.82 TACR1 (0.38) ITGB3ITGA2BCYP19A1ALDH1A1ACHE
SCHEMBL7374011 0.82 DPP4 (0.36) CYP19A1ALDH1A1KDM4EACHE
SCHEMBL7371949 0.81 ACE (0.35) CYP19A1ACEALDH1A1KDM4EACHE
SCHEMBL8621139 0.78 ITGB3 (0.37) ITGB3ITGA2BALDH1A1KDM4EMEN1
SCHEMBL8620398 0.77 MC4R (0.33) CYP19A1ACEALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755374-B1 PROCESS FOR PEPTIDE SEGMENT CONDENSATION MERCK & CO INC (US) 2000-08-16 EP disclosed
EP-0755374-A4 PROCESS FOR PEPTIDE SEGMENT CONDENSATION MERCK & CO INC (US) 1998-09-16 EP disclosed
US-5665882-A Pyridyl ethylation of lactams MERCK & CO., INC. (US) 1997-09-09 US disclosed
EP-0755374-A1 PROCESS FOR PEPTIDE SEGMENT CONDENSATION Merck & Co., Inc. (a New Jersey corp.) (US) 1997-01-29 EP disclosed
WO-1995027727-A2 PROCESS FOR PEPTIDE SEGMENT CONDENSATION MERCK & CO., INC. (US) 1995-10-19 WO disclosed
WO-1995025101-A1 PYRIDIL ETHYLATION OF LACTAMS MERCK & CO., INC. (US) 1995-09-21 WO disclosed