SCHEMBL8619624

SCHEMBL8619624

NCC(N)(C(=O)O)S(=O)(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
MAPT P10636 1/20 0.43
CA9 Q16790 1/20 0.43
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43
SLC1A1 P43005 1/20 0.43
MMP1 P03956 3/20 0.42
HSD11B1 P28845 2/20 0.42
PTPN1 P18031 1/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
EEF2K O00418 1/20 0.40
CNR2 P34972 1/20 0.40
CYP19A1 P11511 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557198 0.82 CA1 (0.49) CA12CA1CA2MAPTCA9
SCHEMBL382142 0.82 SMN1; SMN2 (0.44) CA12CA1CA2MAPTCA9
SCHEMBL7651608 0.82 SMN1; SMN2 (0.44) CA12CA1CA2MAPTCA9
SCHEMBL7372099 0.81 NPC1 (0.45) CA12CA1CA2MAPTCA9
SCHEMBL7372959 0.81 ALDH1A1 (0.45) CA12CA1CA2CA9SLC1A3
SCHEMBL9094518 0.81 CA2 (0.41) CA12CA1CA2CA9SLC1A3
Hydrochloric Acid SCHEMBL382912 0.80 SMN1; SMN2 (0.43) CA12CA1CA2CA9HSD11B1
SCHEMBL7378971 0.77 MMP13 (0.49) CA1CA2MMP1KEAP1NFE2L2
SCHEMBL7452279 0.77 CYP2C9 (0.42) KIF11CA12CA1CA2MAPT
SCHEMBL7375167 0.76 CA2 (0.50) CA12CA1CA2CA9CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832076-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-04-01 EP claimed
WO-1996038426-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-05 WO claimed