SCHEMBL8619928

SCHEMBL8619928

CCCCN(Cc1ccc(C#N)cc1Cl)c1c(NC(C)(C)CC)c(=O)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.37
ABCC8 Q09428 1/20 0.37
KCNJ11 Q14654 1/20 0.37
KCNJ8 Q15842 1/20 0.37
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
P2RX7 Q99572 1/20 0.33
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31
NR1H2 P55055 2/20 0.31
NR1H3 Q13133 2/20 0.31
CYP19A1 P11511 1/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
NR3C1 P04150 1/20 0.31
PGR P06401 1/20 0.31
NR3C2 P08235 1/20 0.31
BCHE P06276 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8621788 0.92 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL7893927 0.82 HTT (0.38) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL7887079 0.82 HTT (0.36) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL4261013 0.78 P2RX7 (0.43) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL8623338 0.76 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL7897114 0.74 HTT (0.37) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL7896906 0.73 HTT (0.39) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL8527319 0.70 P2RX7 (0.39) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL4261010 0.69 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL7898359 0.68 P2RX7 (0.44) ABCC9ABCC8KCNJ11KCNJ8HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US claimed