SCHEMBL8623338

SCHEMBL8623338

CCC(C)(C)Nc1c(NCCCCCc2ccc(C#N)cc2Cl)c(=O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.39
ABCC8 Q09428 1/20 0.39
KCNJ11 Q14654 1/20 0.39
KCNJ8 Q15842 1/20 0.39
P2RX7 Q99572 1/20 0.35
HDAC1 Q13547 1/20 0.35
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
PLK1 P53350 1/20 0.32
TSHR P16473 2/20 0.32
HSD17B10 Q99714 1/20 0.32
EP300 Q09472 3/20 0.31
HAT1 O14929 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4261013 0.85 P2RX7 (0.43) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL7898359 0.76 P2RX7 (0.44) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL8619928 0.76 ABCC9 (0.37) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL4263948 0.75 P2RX7 (0.45) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL7893927 0.73 HTT (0.38) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL4261010 0.72 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL7887079 0.71 HTT (0.36) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL7894054 0.71 ALDH1A1 (0.33) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7596888 0.71 ROCK2 (0.47) P2RX7HDAC1TSHRALDH1A1HTT
SCHEMBL7886987 0.69 P2RX7 (0.39) P2RX7HSD17B10ALDH1A1NPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US disclosed