SCHEMBL8620380

SCHEMBL8620380

COc1cc(OC)c2c(NC(=N)NC=O)cc(-c3ccccc3C)nc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.39
CA9 Q16790 4/20 0.39
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
PDE2A O00408 1/20 0.36
PDE6D O43924 1/20 0.36
PDE6A P16499 1/20 0.36
PDE6G P18545 1/20 0.36
PDE6B P35913 1/20 0.36
PDE6C P51160 1/20 0.36
PDE6H Q13956 1/20 0.36
PDE10A Q9Y233 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 2/20 0.35
POLB P06746 2/20 0.35
MAPT P10636 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618956 0.91 CA12 (0.36) CA2CA9CA12CA1ALDH1A1
SCHEMBL8617297 0.90 CA12 (0.35) CA2CA9CA12CA1ALDH1A1
SCHEMBL8619913 0.88 TGFBR1 (0.39) CA2CA9CA12CA1ALDH1A1
SCHEMBL8618666 0.87 KDM4E (0.44) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL8613210 0.86 KDM4E (0.38) CA2CA9CA12CA1ALDH1A1
SCHEMBL8615214 0.85 PDE2A (0.38) CA2CA9CA12CA1PDE2A
SCHEMBL8620357 0.85 PDE3B (0.38) CA2CA9CA12CA1PDE3B
SCHEMBL8619346 0.84 TACR3 (0.46) CA2CA9CA12CA1ALDH1A1
SCHEMBL8619171 0.83 MAPT (0.39) CA2CA9CA12CA1ALDH1A1
SCHEMBL8617890 0.83 MEN1 (0.45) CA2CA9CA12CA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed