SCHEMBL862066

SCHEMBL862066

Nc1cc(=O)n2ccccc2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.51
ADORA3 P0DMS8 2/20 0.51
ADORA2A P29274 1/20 0.51
ADORA2B P29275 1/20 0.51
ADORA1 P30542 1/20 0.51
PRKDC P78527 1/20 0.51
HPGD P15428 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
MAPT P10636 1/20 0.50
KMT2A Q03164 1/20 0.50
ALDH1A1 P00352 2/20 0.48
GLA P06280 2/20 0.48
GAA P10253 2/20 0.48
HSD17B10 Q99714 2/20 0.48
NPC1 O15118 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
GRM5 P41594 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3958034 0.79 KDM4E (0.55) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL2823070 0.78 KDM4E (0.64) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL12442815 0.78 KDM4E (0.51) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL29918948 0.76 METTL3 (0.54) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL1659994 0.75 KDM4E (0.52) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL28800277 0.75 KDM4E (0.50) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL30132372 0.75 PKM (0.57) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL890517 0.75 KDM4E (0.46) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL31014236 0.75 METTL3 (0.50) KDM4EADORA3ADORA2AADORA2BADORA1
SCHEMBL5132523 0.74 GRIN1 (0.57) KDM4EADORA3ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250002475-A1 PIPERIDINE DERIVATIVES AS METTL3 INHIBITORS EPICS THERAPEUTICS (BE) 2025-01-02 US disclosed
US-12091400-B2 Piperidine derivatives as METTL3 inhibitors EPICS THERAPEUTICS (BE) 2024-09-17 US disclosed
US-20240270716-A1 PIPERIDINE DERIVATIVES AS METTL3 INHIBITORS EPICS THERAPEUTICS (BE) 2024-08-15 US disclosed
US-20240132480-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE TRI-INSTITUTIONAL THERAPEUTICS DISCOVERY INSTITUTE, INC. 2024-04-25 US disclosed
WO-2022150574-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE CORNELL UNIVERSITY (US) 2022-07-14 WO disclosed
EP-1857443-B1 Therapeutic morpholino-substituted compounds ASTRAZENECA AB (SE) 2012-03-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240132480-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE DLD, GCDH, DLAT KDM4E 2390/4885ADORA3 4692/4885ADORA2A 4233/4885
US-20240270716-A1 PIPERIDINE DERIVATIVES AS METTL3 INHIBITORS METTL3, METTL16, DIMT1 KDM4E 872/4885ADORA3 50/4885ADORA2A 139/4885
US-20250002475-A1 PIPERIDINE DERIVATIVES AS METTL3 INHIBITORS METTL3, METTL16, DIMT1 KDM4E 872/4885ADORA3 50/4885ADORA2A 139/4885
US-12091400-B2 Piperidine derivatives as METTL3 inhibitors METTL3, METTL16, DIMT1 KDM4E 872/4885ADORA3 50/4885ADORA2A 139/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.