SCHEMBL8620862

SCHEMBL8620862

COc1cc2nc(-c3ccccc3)cc(C(=O)NC(=N)N)c2cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
HPGD P15428 3/20 0.54
DHODH Q02127 1/20 0.52
TACR3 P29371 2/20 0.52
PLA2G2A P14555 1/20 0.51
MEN1 O00255 7/20 0.51
KMT2A Q03164 7/20 0.51
MAPT P10636 6/20 0.51
KDM4E B2RXH2 6/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
POLB P06746 2/20 0.51
CYP3A4 P08684 2/20 0.50
TP53 P04637 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
LMNA P02545 1/20 0.48
ALOX12 P18054 1/20 0.48
HTT P42858 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CA12 O43570 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8620936 0.87 PLA2G2A (0.69) TACR3PLA2G2AMEN1KMT2AMAPT
SCHEMBL8617885 0.86 CA2 (0.49) ALDH1A1HPGDDHODHTACR3MEN1
SCHEMBL8616493 0.86 TACR3 (0.71) ALDH1A1HPGDTACR3PLA2G2AMEN1
SCHEMBL8614842 0.86 DHODH (0.72) ALDH1A1HPGDDHODHMEN1KMT2A
SCHEMBL8619812 0.84 ALDH1A1 (0.54) ALDH1A1HPGDDHODHPLA2G2AMEN1
SCHEMBL8613185 0.84 PDE10A (0.49) ALDH1A1HPGDTACR3MEN1KMT2A
SCHEMBL8617709 0.83 PDE10A (0.69) ALDH1A1HPGDDHODHMEN1KMT2A
SCHEMBL8620626 0.83 ALDH1A1 (0.48) ALDH1A1HPGDDHODHPLA2G2AMEN1
SCHEMBL8617743 0.83 CYP3A4 (0.65) ALDH1A1HPGDDHODHTACR3MEN1
SCHEMBL8613846 0.83 KDM4E (0.67) ALDH1A1MEN1KMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed