SCHEMBL8620971

SCHEMBL8620971

O=C(OC(=O)C1Cc2ccccc2CN1C(=O)O)C1Cc2ccccc2CN1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 3/20 0.47
ACE P12821 4/20 0.47
POLB P06746 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PREP P48147 2/20 0.43
CHEK1 O14757 1/20 0.43
JAK2 O60674 1/20 0.43
LMNA P02545 2/20 0.42
PKM P14618 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MMP3 P08254 1/20 0.40
MMP8 P22894 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908771 0.85 ACE (0.61) ACEPOLBTDP1L3MBTL1CHEK1
SCHEMBL4573235 0.85 ACE (0.61) ACEPOLBTDP1L3MBTL1CHEK1
SCHEMBL3840630 0.85 ACE (0.61) ACEPOLBTDP1L3MBTL1CHEK1
SCHEMBL28561301 0.82 ACE (0.48) ACEPOLBTDP1L3MBTL1PREP
SCHEMBL4480032 0.79 NR1D1 (0.49) NR1D1ACEPOLBTDP1L3MBTL1
SCHEMBL4627296 0.77 ACE (0.60) ACEPOLBTDP1L3MBTL1CHEK1
SCHEMBL5720519 0.77 ACE (0.60) ACEPOLBTDP1L3MBTL1CHEK1
SCHEMBL25377457 0.77 PREP (0.69) PREP
SCHEMBL3891147 0.77 TACR1 (0.47) NR1D1ACEPOLBTDP1L3MBTL1
SCHEMBL25349861 0.77 TACR1 (0.47) NR1D1ACEPOLBTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-10291979-A None JP disclosed
JP-H10291979-A PRODUCTION OF 1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACID TERTIARY BUTYL AMIDE ICHIKAWA GOSEI KAGAKU KK 1998-11-04 JP disclosed