SCHEMBL8621045

SCHEMBL8621045

CN(C)CCOc1cc2c(cc1I)CCN2

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.37
HTR7 P34969 3/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.33
HTR1B P28222 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
PARP1 P09874 2/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
ROCK2 O75116 1/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7756067 0.83 MAPT (0.40) HRH3HTR7KDM4EMAPTTHRA
SCHEMBL7752192 0.83 HTR7 (0.42) HRH3HTR7BCHEACHE
SCHEMBL8612335 0.83 HTR7 (0.44) HRH3HTR7KDM4EMAPTHTR1B
SCHEMBL8615260 0.82 NOS3 (0.39) HRH3HTR7KDM4EMAPTHTR1B
SCHEMBL8389373 0.76 HTR7 (0.40) HRH3HTR7KDM4EMAPTTHRB
SCHEMBL15880025 0.74 HRH3 (0.58) HRH3KDM4EPARP1
SCHEMBL8619296 0.73 SLC6A4 (0.38) HRH3KDM4EMAPTTHRBPARP1
SCHEMBL9098005 0.73 NR4A2 (0.51) HRH3HTR7KDM4EHTR1B
SCHEMBL14842640 0.69 HTR1B (0.48) HTR7KDM4EHTR1BDRD2DRD1
SCHEMBL1572695 0.68 CYP1A2 (0.54) HRH3HTR7KDM4EHTR1BTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed