SCHEMBL8622258

SCHEMBL8622258

Cc1cccc(OCc2ccccc2CCl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.47
TP53 P04637 1/20 0.46
POLB P06746 1/20 0.46
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
ACHE P22303 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KMT2A Q03164 1/20 0.43
MAOA P21397 1/20 0.43
KDM4E B2RXH2 1/20 0.43
CCNB2 O95067 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1548999 0.91 MAOB (0.54) MAOBTP53POLBDRD2DRD4
SCHEMBL13794364 0.86 MAOB (0.50) MAOBTP53POLBDRD2DRD4
SCHEMBL8618327 0.86 GRM5 (0.39) MAOBRAB9AKMT2AMAOA
SCHEMBL257758 0.83 NR4A2 (0.60) MAOBTP53POLBDRD2DRD4
SCHEMBL12183099 0.83 CCNB2 (0.58) MAOBTP53POLBDRD2DRD4
SCHEMBL1539409 0.81 LMNA (0.50) MAOBTP53DRD2DRD4NPC1
SCHEMBL25128164 0.80 ALDH1A1 (0.54) MAOBTP53POLBDRD2DRD4
SCHEMBL2290158 0.80 MAOB (0.54) MAOBTP53POLBDRD2DRD4
SCHEMBL21084234 0.80 LMNA (0.57) MAOBRAB9AMAPTHTTTSHR
SCHEMBL8623315 0.80 POLB (0.47) MAOBTP53POLBDRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0658541-B1 PROCESS FOR PRODUCING CARBOXYLIC ACID DERIVATIVE SHIONOGI & CO (JP) 1998-05-20 EP disclosed
US-5510506-A Process for producing carboxylic acid derivatives SHIONOGI & CO., LTD. (JP) 1996-04-23 US disclosed
EP-0658541-A1 PROCESS FOR PRODUCING CARBOXYLIC ACID DERIVATIVE SHIONOGI & CO., LTD. (JP) 1995-06-21 EP disclosed