SCHEMBL8622671

SCHEMBL8622671

CN(C)CCn1ccc2cc(NC(=O)NC3=c4ccccc4=C(c4ccccn4)CC3)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.43
EGFR P00533 5/20 0.41
PIK3CA P42336 1/20 0.40
MTOR P42345 1/20 0.40
HTR2C P28335 3/20 0.40
HTR2B P41595 2/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C19 P33261 1/20 0.39
RECQL P46063 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HTR2A P28223 1/20 0.38
ALOX5 P09917 1/20 0.37
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622676 0.80 HTR2B (0.51) HTR6EGFRPIK3CAMTORHTR2C
SCHEMBL6714734 0.73 HTR6 (0.54) HTR6HTR2CHTR2A
SCHEMBL6719408 0.70 HDAC3 (0.52) HTR6HTR2CMAPTHTR2A
SCHEMBL8710351 0.67 MAPT (0.62) HTR2CHTR2BKDM4EMEN1TP53
SCHEMBL7258134 0.65 HTR1D (0.67) HTR6HTR2CHTR2A
SCHEMBL21671857 0.65 HTR6 (0.58) HTR6EGFRHTR2CHTR2A
SCHEMBL9400613 0.65 HTR2B (0.65) HTR2CHTR2BKDM4EMEN1TP53
SCHEMBL18960579 0.64 HTR2C (0.56) HTR6HTR2CCYP1A2CYP2D6HTR2A
SCHEMBL8615090 0.64 HTR6 (0.49) HTR6PIK3CAMTORHTR2CHTR2B
SCHEMBL9400583 0.64 MEN1 (0.73) HTR2CHTR2BKDM4EMEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998047868-A1 HETEROCYCLE-CONTAINING UREA DERIVATIVES AS 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-10-29 WO disclosed