SCHEMBL8622975

SCHEMBL8622975

BrCc1cccc(C=Cc2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
TRPA1 O75762 1/20 0.52
TSHR P16473 1/20 0.52
NFE2L2 Q16236 5/20 0.50
MAOB P27338 3/20 0.50
CYP19A1 P11511 2/20 0.50
MAOA P21397 2/20 0.50
LCK P06239 1/20 0.49
RELA Q04206 1/20 0.45
HDAC4 P56524 1/20 0.42
MEF2D Q14814 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622972 1.00 ALDH1A1 (0.52) ALDH1A1TRPA1TSHRNFE2L2MAOB
SCHEMBL9454709 1.00 ALDH1A1 (0.52) ALDH1A1TRPA1TSHRNFE2L2MAOB
SCHEMBL26316674 0.85 NFE2L2 (0.56) ALDH1A1NFE2L2CYP19A1LCKRELA
SCHEMBL7489498 0.82 ALDH1A1 (0.39) ALDH1A1TRPA1TSHRNFE2L2LCK
SCHEMBL27450402 0.82 ALDH1A1 (0.39) ALDH1A1TRPA1TSHRNFE2L2MAOB
SCHEMBL18197883 0.82 ALDH1A1 (0.39) ALDH1A1TRPA1TSHRNFE2L2LCK
SCHEMBL7489493 0.82 ALDH1A1 (0.39) ALDH1A1TRPA1TSHRNFE2L2LCK
SCHEMBL3565889 0.81 KDM4E (0.59) ALDH1A1TSHRHDAC4MEF2DKDM4E
SCHEMBL3565886 0.81 KDM4E (0.59) ALDH1A1TSHRHDAC4MEF2DKDM4E
SCHEMBL9455094 0.81 RAB9A (0.45) ALDH1A1TRPA1TSHRNFE2L2LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719303-A USEFUL FOR MEDICALLY TREATING HYPERLIPEMIA EISAI CO., LTD. (JP) 1998-02-17 US disclosed
EP-0688325-A1 PHOSPHONIC ACID DERIVATIVES Eisai Co., Ltd. (JP) 1995-12-27 EP disclosed
WO-1994020508-A1 PHOSPHONIC ACID DERIVATIVES EISAI CO., LTD. (JP) 1994-09-15 WO disclosed
US-5234946-A Anticholesterol, antilipemic BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-10 US disclosed
EP-0318860-B1 SUBSTITUTED ALKYLAMINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-16 EP disclosed
EP-0318860-A2 Substituted alkylamine derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1989-06-07 EP disclosed
EP-0007576-B1 ESTERS OF STILBENE DERIVATIVES, PROCESS FOR THEIR PREPARATION, STILBENE-ALCOHOLS AS INTERMEDIATE PRODUCTS, USE OF THE ESTERS AS INSECTICIDES BAYER AG (DE) 1983-11-16 EP disclosed
US-4271186-A Stilbene compounds and insecticidal/acaricidal compositions BAYER AKTIENGESELLSCHAFT (DE) 1981-06-02 US disclosed
EP-0007576-A2 Esters of stilbene derivatives, process for their preparation, stilbene-alcohols as intermediate products, use of the esters as insecticides BAYER AG (DE) 1980-02-06 EP disclosed