SCHEMBL8625170

SCHEMBL8625170

CCn1cc(C(=O)O)c(=O)c2c(Cl)c(F)ccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.52
HPGD P15428 6/20 0.52
HSD17B10 Q99714 5/20 0.52
ALDH1A1 P00352 5/20 0.52
TSHR P16473 3/20 0.52
RAB9A P51151 1/20 0.52
CHRM1 P11229 3/20 0.48
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
APEX1 P27695 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
DRD3 P35462 1/20 0.46
LMNA P02545 5/20 0.46
HTT P42858 3/20 0.46
PIK3CG P48736 2/20 0.46
PIK3CD O00329 1/20 0.46
PIK3R1 P27986 1/20 0.46
PIK3CA P42336 1/20 0.46
POLB P06746 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627262 0.86 ALDH1A1 (0.54) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL9321178 0.79 KDM4E (0.49) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL9148727 0.79 LMNA (0.51) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL14845181 0.77 KDM4E (0.55) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL8483940 0.77 ALDH1A1 (0.61) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL15999507 0.76 KDM4E (0.49) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL8111305 0.76 FOXO1 (0.52) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL14845200 0.76 FOXO1 (0.52) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL15999546 0.76 KDM4E (0.54) KDM4EHPGDHSD17B10ALDH1A1TSHR
SCHEMBL1366635 0.76 KDM4E (0.68) KDM4EHPGDHSD17B10ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684942-B1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORP (US) 1998-06-10 EP disclosed
EP-0684942-A4 1995-12-27 EP disclosed
EP-0684942-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1995-12-06 EP disclosed
US-5430152-A Heating aminoarylester in presence of chlorosulfonic acid, oleum HOECHST CELANESE CORPORATION (US) 1995-07-04 US disclosed
WO-1994019312-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1994-09-01 WO disclosed