SCHEMBL8627264

SCHEMBL8627264

COc1cc[c]c(C=S)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
CA7 P43166 3/20 0.34
CA9 Q16790 3/20 0.34
CA12 O43570 2/20 0.34
CA14 Q9ULX7 2/20 0.34
CYP1A2 P05177 5/20 0.34
CYP1A1 P04798 3/20 0.34
CYP1B1 Q16678 3/20 0.34
ALDH1A1 P00352 3/20 0.33
ACHE P22303 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP3A4 P08684 2/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1637725 0.80 ALDH1A1 (0.44) CA1CA2CA7CA9CA12
SCHEMBL15066961 0.76 ALDH1A1 (0.41) CA1CA2CA7CA9CA12
SCHEMBL10695354 0.73 TRPA1 (0.55) CYP1A2CYP1A1CYP1B1ALDH1A1CYP3A4
SCHEMBL1569519 0.72
SCHEMBL7380255 0.72 THRB (0.51) CA1CA2CA7CA9CA12
SCHEMBL7380258 0.72 THRB (0.51) CA1CA2CA7CA9CA12
SCHEMBL5871896 0.71 MAPT (0.42) ALDH1A1HPGDMEN1MAPTKMT2A
SCHEMBL160135 0.70
SCHEMBL77754 0.70 CA1 (0.39) CA1CA2CA7CA9CA12
SCHEMBL10897682 0.70 KMT2A (0.40) CA1CA2CA9CA12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5795905-A 3-AMINO-5-PHENYL-1,2,4-TRIAZOLES NEUROCRINE BIOSCIENCES, INC. (US) 1998-08-18 US claimed
EP-0846108-A1 AMINO-SUBSTITUTED THIADIAZOLES, PYRIMIDINES, TRIAZINES OR TRIAZOLES USEFUL AS CTF RECEPTOR ANTAGONISTS NEUROCRINE BIOSCIENCES, INC. (US) 1998-06-10 EP claimed
WO-1996039400-A1 AMINO-SUBSTITUTED THIADIAZOLES, PYRIMIDINES, TRIAZINES OR TRIAZOLES USEFUL AS CTF RECEPTOR ANTAGONISTS NEUROCRINE BIOSCIENCES, INC. (US) 1996-12-12 WO claimed