SCHEMBL8627552

SCHEMBL8627552

NS(=O)(=O)c1ccc(-c2nn[c]n2-c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.50
CA1 P00915 10/20 0.49
CA2 P00918 10/20 0.49
CA12 O43570 6/20 0.49
CA9 Q16790 6/20 0.49
CA4 P22748 1/20 0.47
CA7 P43166 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
PTGS1 P23219 3/20 0.46
CA5A P35218 1/20 0.44
CA5B Q9Y2D0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633825 0.76 CA2 (0.48) PTGS2CA1CA2CA12CA9
SCHEMBL8628934 0.75 HSD17B10 (0.44)
SCHEMBL8631163 0.70 KDM4E (0.40) PTGS2
SCHEMBL8629241 0.69 CA2 (0.40) PTGS2CA1CA2CA12CA9
SCHEMBL308881 0.68 CA2 (1.00) PTGS2CA1CA2CA12CA9
SCHEMBL6482321 0.68 CA2 (1.00) PTGS2CA1CA2CA12CA9
SCHEMBL497671 0.68 PTGS2 (0.81) PTGS2CA1CA2CA12CA9
Hydrochloric Acid SCHEMBL30685243 0.66 CA2 (0.95) PTGS2CA1CA2CA12CA9
SCHEMBL5594366 0.66 PTGS2 (0.90) PTGS2PTGS1
SCHEMBL795390 0.66 AVPR1A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4399131-A Cephem derivatives HOECHST AG (DE) 1983-08-16 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed