SCHEMBL8629241

SCHEMBL8629241

C=CCn1[c]nnc1-c1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 14/20 0.40
CA9 Q16790 13/20 0.40
CA12 O43570 12/20 0.40
CA1 P00915 10/20 0.40
CA7 P43166 2/20 0.40
CA5A P35218 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
PTGS2 P35354 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8626448 0.78 L3MBTL1 (0.45)
SCHEMBL8633825 0.74 CA2 (0.48) CA2CA9CA12CA1CA7
SCHEMBL8625324 0.73 CA2 (0.40) CA2CA9CA12CA1CA7
SCHEMBL8627552 0.69 PTGS2 (0.50) CA2CA9CA12CA1CA7
SCHEMBL4605045 0.60 CA2 (0.57) CA2CA9CA12CA1CA7
SCHEMBL202948 0.59 CA2 (0.81) CA2CA9CA12CA1CA7
Ammonia Solution, Strong SCHEMBL9404175 0.59 CA2 (0.55) CA2CA9CA12CA1CA7
SCHEMBL8628373 0.59 CA2 (0.51) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL992952 0.59 CA2 (0.90) CA2CA9CA12CA1CA7
SCHEMBL1698660 0.58 CA2 (0.60) CA2CA9CA12CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4399131-A Cephem derivatives HOECHST AG (DE) 1983-08-16 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed