SCHEMBL8633825

SCHEMBL8633825

Cn1[c]nnc1-c1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.48
CA9 Q16790 12/20 0.48
CA12 O43570 11/20 0.48
CA1 P00915 9/20 0.48
PTGS2 P35354 7/20 0.46
CA5A P35218 3/20 0.44
CA5B Q9Y2D0 3/20 0.44
CA3 P07451 1/20 0.44
CA6 P23280 1/20 0.44
CA7 P43166 1/20 0.44
CA4 P22748 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627552 0.76 PTGS2 (0.50) CA2CA9CA12CA1PTGS2
SCHEMBL8629241 0.74 CA2 (0.40) CA2CA9CA12CA1PTGS2
SCHEMBL8628373 0.71 CA2 (0.51) CA2CA9CA12CA1PTGS2
SCHEMBL12692373 0.67 CA12 (0.86) CA2CA9CA12CA1PTGS2
SCHEMBL202948 0.65 CA2 (0.81) CA2CA9CA12CA1CA5A
SCHEMBL11623852 0.65 PTGS2 (0.66) PTGS2
SCHEMBL2605787 0.65 CA1 (1.00) CA2CA9CA12CA1PTGS2
P-Toluenesulfonamide SCHEMBL31527821 0.64 CA2 (1.00) CA2CA9CA12CA1PTGS2
P-Toluenesulfonamide SCHEMBL7370 0.64 CA2 (1.00) CA2CA9CA12CA1PTGS2
P-Toluenesulfonamide SCHEMBL1331323 0.64 CA2 (1.00) CA2CA9CA12CA1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4399131-A Cephem derivatives HOECHST AG (DE) 1983-08-16 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed