SCHEMBL8627772

SCHEMBL8627772

COc1ccc(-c2c[nH]nc2-c2ccccc2S(N)(=O)=O)cc1C

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.47
PTGS1 P23219 5/20 0.47
BRD4 O60885 1/20 0.42
P2RX3 P56373 4/20 0.40
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CA4 P22748 1/20 0.38
F10 P00742 2/20 0.38
F2 P00734 1/20 0.37
PTGES2 Q9H7Z7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630031 0.88 PTGS2 (0.41) PTGS2PTGS1CA12CA2CA9
SCHEMBL8629321 0.88 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL8628069 0.86 F10 (0.35) PTGS2PTGS1F10PTGES2
SCHEMBL7780829 0.85 PTGS2 (0.62) PTGS2PTGS1CA12CA2CA9
SCHEMBL8632812 0.83 ALOX5AP (0.47) PTGS2PTGS1F10
SCHEMBL8632216 0.82 SCN9A (0.46) F10F2
SCHEMBL8632840 0.82 LRRK2 (0.42) PTGS2PTGS1CA12CA2CA9
SCHEMBL8631346 0.81 NPC1 (0.40) CA2PTGES2
SCHEMBL8627632 0.79 CA1 (0.42) CA12CA2CA9CA4
SCHEMBL8632289 0.79 AKR1B1 (0.40) PTGS2CA12CA2CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed