SCHEMBL8628053

SCHEMBL8628053

CS(=O)(=O)c1ccc(-n2ncc(-c3ccc(NC(=O)C(F)(F)F)cc3)c2C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
PTGS2 P35354 10/20 0.43
PTGS1 P23219 2/20 0.43
EPHX2 P34913 2/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.40
TRPC1 P48995 1/20 0.40
TRPC3 Q13507 1/20 0.40
STIM1 Q13586 1/20 0.40
ORAI1 Q96D31 1/20 0.40
STIM2 Q9P246 1/20 0.40
DPP4 P27487 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629371 0.81 PTGS2 (0.52) PTGS2PTGS1EPHX2CYP2C9
SCHEMBL8631359 0.78 MELK (0.63) KMT2ACA12CA1CA2CA9
SCHEMBL18850964 0.76 CA12 (0.70) KMT2ACA12CA1CA2CA9
SCHEMBL8633742 0.73 POLB (0.55) KMT2APTGS2PTGS1MAPT
SCHEMBL2859374 0.73 MAPT (0.52) CA1CA2CA9PTGS2PTGS1
SCHEMBL8631118 0.72 MAPT (0.45) KMT2ACA1CA2CA9PTGS2
SCHEMBL7772921 0.72 CA12 (0.47) KMT2ACA12CA1CA2CA9
SCHEMBL8631115 0.70 KMT2A (0.49) KMT2ACA1CA2CA9PTGS2
SCHEMBL8955949 0.68 PTGS2 (0.77) PTGS2PTGS1CYP2C9
SCHEMBL7777513 0.68 CA12 (0.45) KMT2ACA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed